僅用于工業(yè)應(yīng)用或科學(xué)研究,不可用于人類或動(dòng)物的臨床診斷或治療,非藥用.Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediatated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59±0.07 and 0.516±0.065 μM and IC50 of 1.58 and 3.29 μM, respectively.Stiripentol (STP) 是一種抗驚厥劑,其可以抑制由 CYP3A4 (非競(jìng)爭(zhēng)性) 和 CYP2C19 (競(jìng)爭(zhēng)性地) 介導(dǎo)的 CLB 向 N-desmethylclobazam (NCLB) 的 N-去甲基化,其 Ki 值分別為 1.59±0.07 和 0.516±0.065 μM,IC50 值分別為 1.58 和 3.29 μM